Basic Peptide Information

DICL ID
DICL_Pep_06220
Ion Channel
Neuronal acetylcholine receptor subunit alpha-2/beta-4
Peptide Function
Antagonist
Gene Name
CHRNA2/CHRNB4

Activity Data (nM)

IC50
>10000 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
GCCSHPVCKAMSPIC
Peptide UniProt Accession
Not available
UniParc
UPI0034A632A2
Peptide Synonyms/Alias
[CHEMBL4215824; BDBM50459652]
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available

Experimental Conditions

pH
Not mention
Holding Potential (mV)
−70 mV
Temperature
Room Temperature
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available